Tirzep (UPZEP) 30mg Vial

UpZep 30mg is a groundbreaking injectable peptide that work by enhancing insulin secretion, decrease glucagon levels, slow gastric emptying, and increase satiety—making it highly effective for reducing body weight and improving glucose metabolism.

By engaging two powerful incretin pathways, UpZep 30mg provides superior results in appetite regulation and fat loss. It also supports improvements in cardiovascular markers, blood sugar control, and inflammation.

Because UpZep 30mg comes in powdered form, it requires reconstitution prior to injection. Once prepared, it is injected subcutaneously once weekly, with dosage gradually increased to reduce the risk of side effects.

Benefits

• Promotes significant and sustained fat loss

• Suppresses appetite and food cravings

• Improves insulin sensitivity and blood glucose regulation

• Enhances satiety and delays gastric emptying

• Supports long-term weight management and metabolic health

• Once-weekly administration for convenience

Side effects
While UpZep 30mg is generally well tolerated, users may experience:

• Nausea, especially during dose escalation

• Bloating or digestive discomfort

• Constipation or diarrhea

• Headache or fatigue

• Injection site irritation (mild)

• Rarely, dizziness or low blood sugar in sensitive individuals

These effects are typically dose-dependent and improve as the body adjusts. Slow titration is recommended.

Dosages & Protocol
Starting dose: 2.5mg once weekly for 2–4 weeks
Titration: Increase to 5mg weekly, then gradually to 10mg, 12.5mg, or 15mg as tolerated
Maximum dose: 15mg once per week for advanced metabolic or weight-loss goals
Cycle Duration: Can be used long-term (3–6 months or more) for weight loss and insulin resistance reversal

PLEASE MAKE USE OF OUR PEPTIDE CALCULATOR FOR FURTHER DOSAGE GUIDANCE.

How to administer – reconstitution and how to inject
UpZep 30mg comes as a lyophilized powder in a single vial, with one amp of bacteriostatic water included

Reconstitution:

• Reconstitute with 1ml or 2ml of bacteriostatic water, depending on your preferred concentration

• Inject the water slowly down the side of the vial

• Swirl gently until fully dissolved—do not shake

Injection:

• Use a U100 insulin syringe (29–31 gauge)

• Dosages (if reconstituted with 2ml bacteriostatic water):

  • 2.5mg = 16.5 units – week 1 

  • 5mg = 33 units – week 2 & 3

  • 7.5mg = 50 units – week 4 & maintenance 

• Inject subcutaneously into the abdomen, thigh, or upper arm once per week

• Clean the injection site with an alcohol swab prior to inecting

• Rotate injection sites weekly to prevent irritation

Storage
After reconstitution: store refrigerated at 2–8°C and use within 30 days

Half life & detectability
Half-Life: Approximately 5 days, allowing for once-weekly dosing
Detection Time: Not commonly screened in routine drug testing, but detection is possible through advanced metabolic/hormonal analysis
For athletes subject to drug testing, it is important to consider these detection times and plan accordingly to avoid positive tests for banned substances.