Ketotifen – Zaditen 1mg is primarily an anti-allergic medication that blocks histamine receptors and prevents the release of inflammatory substances from mast cells. It is commonly prescribed for conditions such as asthma, hay fever, and chronic allergic symptoms. However, in the performance-enhancing and fat-loss community, Ketotifen has gained popularity for its ability to upregulate beta-2 adrenergic receptors, which are often desensitized by prolonged use of stimulants like Clenbuterol.
By resetting these receptors, Ketotifen allows users to maintain the effectiveness of fat-burning compounds without the need for off-cycles. It also improves sleep quality and reduces systemic inflammation.
Benefits
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Reduces allergic symptoms like itching, hives, and asthma
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Prevents beta-2 receptor downregulation during Clenbuterol use
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Prolongs the effectiveness of stimulants in fat-loss protocols
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Improves sleep quality
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Mild sedative effects which can aid rest and recovery
Side effects
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Drowsiness or sedation, especially at the beginning of use
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Dry mouth
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Increased appetite or slight weight gain in some individuals
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Dizziness
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Mild gastrointestinal discomfort
Dosages & Protocol
Dosages for Men and Women:
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Standard dose: 1mg once or twice daily
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When used to maintain Clenbuterol effectiveness: 1mg before bed is common
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Start with 1mg nightly and adjust based on tolerance
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Cycle length: Can be used throughout Clenbuterol cycles or up to several weeks continuously
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Avoid alcohol or other sedatives when using due to additive drowsiness
How to administer
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Take orally with water
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Best taken in the evening due to potential sedative effects
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May be taken with or without food
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Do not drive or operate machinery until you know how it affects you
Storage
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Store in a cool, dry place below 25°C
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Keep the packet tightly closed and away from moisture and heat
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Keep out of reach of children
Half-life & detectability
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Half-life: Approximately 12 hours, allowing once-daily dosing
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Detection time: Not typically screened for in drug testing; not a banned substance
For athletes subject to drug testing, it is crucial to consider these detection times to avoid positive tests for banned substances.
